BDBM50607604 CHEMBL5219712

SMILES CNC(=O)c1cccc(c1)CNC(=O)[C@H]2CCCN2C(=O)C3(CCCC3)c4ccc(cc4)Cl

InChI Key InChIKey=FKSCOWJURPRAGR-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50607604   

TargetHistone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607604(CHEMBL5219712)
Affinity DataIC50: 10nMAssay Description:Inhibition of full-length P300 (unknown origin) using ARTKQTARKSTGGKAPRKQLAGG-K(Biotin)-amide as substrate preincubated for 60 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed