BDBM50608806 CHEMBL5284816

SMILES CC(C)C(C(C)NC(=O)Nc1ccc(Br)cc1)C(O)=O

InChI Key InChIKey=GYDLWCFVSYYOGO-UHFFFAOYSA-N

Data  8 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50608806   

TargetfMet-Leu-Phe receptor(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  51nMAssay Description:Agonist activity at FPR1 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  13nMAssay Description:Agonist activity at FPR1 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  98nMAssay Description:Agonist activity at FPR1 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at FPR1 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetN-formyl peptide receptor 2(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  855nMAssay Description:Agonist activity at FPR2 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetN-formyl peptide receptor 2(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  3.24E+3nMAssay Description:Agonist activity at FPR2 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetN-formyl peptide receptor 2(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  9.94E+3nMAssay Description:Agonist activity at FPR2 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetN-formyl peptide receptor 2(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50608806(CHEMBL5284816)
Affinity DataEC50:  25nMAssay Description:Agonist activity at FPR2 (unknown origin) expressed in CHO/Galpha16 cells assessed as increase in calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed