BDBM50608962 CHEMBL5288169

SMILES Cc1cc2nc(CCc3nc4nc(C)cc(C)n4n3)cc(O)n2n1

InChI Key InChIKey=MWQJNCZLMGLERH-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50608962   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Nirma University

Curated by ChEMBL

LigandBDBM50608962(CHEMBL5288169)Copy SMILESCopy InChI

Affinity DataIC50: 44nMAssay Description:Inhibition of human PDE10A (449 to 789 residues) expressed in Escherichia coli BL21(DE3) using cAMP as substrate incubated for 30 mins by HTRF analys...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
4/20/2024
Entry Details
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