BDBM50652597 CHEMBL5639286

SMILES COc1ccc(COc2ccc(Cn3cnc4cc(C(=O)N5CC6(COC6)C5)cnc43)cc2OC)cn1

InChI Key

PDB links: 1 PDB ID matches this monomer.

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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50652597   

LigandPNGBDBM50652597(CHEMBL5639286)
Affinity DataIC50: 15nMAssay Description:Inhibition of N-terminal GST-fused human CSF1R (538 to 972 residues) expressed in Sf21 insect cells preincubated for 15 mins followed by substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
LigandPNGBDBM50652597(CHEMBL5639286)
Affinity DataIC50: 40nMAssay Description:Inhibition of human CSF1R phosphorylation in CSF1-stimulated HEK293 cells by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed