BDBM50652599 CHEMBL5642438

SMILES COc1ccc(COc2ccc(Cn3cnc4cc(C#N)cnc43)cc2OC)cn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50652599   

LigandPNGBDBM50652599(CHEMBL5642438)
Affinity DataIC50: 125nMAssay Description:Inhibition of N-terminal GST-fused human CSF1R (538 to 972 residues) expressed in Sf21 insect cells preincubated for 15 mins followed by substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
LigandPNGBDBM50652599(CHEMBL5642438)
Affinity DataIC50: 204nMAssay Description:Inhibition of human CSF1R phosphorylation in CSF1-stimulated HEK293 cells by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed