BDBM507386 US11046680, Example 265.0::US11046680, Example 266.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc(-c2ccn(C)n2)n1-c1c(OC)cccc1OC)c1ccc(cc1C#N)C#N

InChI Key InChIKey=SUVNHFSVINBRKE-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 507386   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM507386(US11046680, Example 266.0 | US11046680, Example 26...)
Affinity DataEC50:  0.400nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM507386(US11046680, Example 266.0 | US11046680, Example 26...)
Affinity DataEC50:  70nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent