BDBM507501 US11046680, Example 380.0

SMILES CO[C@@H](CS(=O)(=O)Nc1nnc(-c2ccn(C)n2)n1-c1c(OC)cccc1OC)c1ccc(Cl)cc1S(C)(=O)=O

InChI Key InChIKey=ZYJBKAFWIZYRAT-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 507501   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM507501(US11046680, Example 380.0)
Affinity DataEC50:  0.400nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent