BDBM519446 (4S,5R)-5-(3-fluoro-5-(trifluoromethyl)phenyl)-4-methyl-3-(3-(6-methyl-2,3-dihydro-4H-pyrido[3,2-b][1,4]oxazin-4- yl)propanoyl)oxazolidin-2-one::US11141410, Example 92

SMILES C[C@H]1[C@H](OC(=O)N1C(=O)CCN1CCOc2ccc(C)nc12)c1cc(F)cc(c1)C(F)(F)F

InChI Key InChIKey=FIJVUPDPGAZWSS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 519446   

TargetN-acetylglucosamine-1-phosphotransferase subunits alpha/beta(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM519446((4S,5R)-5-(3-fluoro-5-(trifluoromethyl)phenyl)-4-m...)
Affinity DataIC50: 240nMAssay Description:The TarO biochemical enzymatic assay is a liquid chromatography-mass spectroscopy (LC-MS) based end point assay that measures C55-P-P-GlcNAc (LIPID I...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2022
Entry Details
US Patent