BDBM521470 (R)-N-(1-(2- Methyl-4- ((3-methyl- [1,1'- biphenyl]- 4-yl)methyl) piperazine- 1-carbonyl)- 1H-pyrazol-3- yl)acetamide::US11149037, Example 208

SMILES C[C@@H]1CN(Cc2ccc(cc2C)-c2ccccc2)CCN1C(=O)n1ccc(NC(C)=O)n1

InChI Key InChIKey=WYIIEHSHESASLM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 521470   

TargetMonoglyceride lipase(Human)
H. Lundbeck

US Patent
LigandPNGBDBM521470((R)-N-(1-(2- Methyl-4- ((3-methyl- [1,1'- biphenyl...)
Affinity DataIC50: 100nMAssay Description:Proteomes (mouse brain membrane fraction or cell lysates for mouse assays; human prefrontal cortex or PC3 cell membrane fractions for human assays) (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent