BDBM521474 US11149040, Example 4.0::US11149040, Example 5.0

SMILES COC[C@@H]1COc2ccccc2-c2nnc(NS(=O)(=O)[C@@H](C)[C@@H](OC(C)C)c3ncc(C)cn3)n12

InChI Key InChIKey=RPICFLKUIPGMFC-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 521474   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM521474(US11149040, Example 5.0 | US11149040, Example 4.0)
Affinity DataEC50:  17nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM521474(US11149040, Example 5.0 | US11149040, Example 4.0)
Affinity DataEC50:  130nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent