BDBM521488 US11149040, Example 18.0::US11149040, Example 19.0

SMILES COc1ccc2OC[C@@H](CO)n3c(NS(=O)(=O)[C@@H](C)[C@@H](OC(C)C)c4ncc(C)cn4)nnc3-c2n1

InChI Key InChIKey=VLQYNAIZPBCOMK-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 521488   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM521488(US11149040, Example 19.0 | US11149040, Example 18....)
Affinity DataEC50:  640nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM521488(US11149040, Example 19.0 | US11149040, Example 18....)
Affinity DataEC50:  990nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent