BDBM521504 US11149040, Example 34.0::US11149040, Example 35.0

SMILES COC[C@@H]1COc2ncccc2-c2nnc(NS(=O)(=O)CCc3ncc(C)cn3)n12

InChI Key InChIKey=LDTOSJFLJUMRFJ-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 521504   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM521504(US11149040, Example 35.0 | US11149040, Example 34....)
Affinity DataEC50:  180nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM521504(US11149040, Example 35.0 | US11149040, Example 34....)
Affinity DataEC50:  180nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent