BDBM523786 US11136312, Compound AH.2.126

SMILES Fc1ccc2[nH]c(cc2c1)-c1nnc(SCc2ccccc2)n1CCCc1c[nH]cn1

InChI Key InChIKey=VYCZFTGUPKITKZ-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 523786   

TargetSomatostatin receptor type 4(Human)
Board of Trustees of The Southern Illinois University

US Patent
LigandPNGBDBM523786(US11136312, Compound AH.2.126)
Affinity DataKi:  776nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetSomatostatin receptor type 3(Human)
Board of Trustees of The Southern Illinois University

US Patent
LigandPNGBDBM523786(US11136312, Compound AH.2.126)
Affinity DataEC50:  1.13E+3nMAssay Description:Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetSomatostatin receptor type 2(Human)
Board of Trustees of The Southern Illinois University

US Patent
LigandPNGBDBM523786(US11136312, Compound AH.2.126)
Affinity DataKi: >1.00E+4nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent