BDBM524156 US11166942, Compound 58

SMILES O[C@@H](COc1ccc(Cl)c(F)c1)CN1CCN(CC1)NC(=O)c1ccc2cc(Cl)ccc2n1

InChI Key InChIKey=OOHNNNJXHAZGCG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 524156   

TargetCyclic AMP-dependent transcription factor ATF-4(Human)
Praxis Biotech

US Patent
LigandPNGBDBM524156(US11166942, Compound 58)
Affinity DataIC50: 5.70nMAssay Description:The ATF4 reporter was prepared by fusing the human full length 5′UTR of ATF4 (NCBI Accession No. BC022088.2) upstream of the firefly luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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