BDBM527746 US11186590, Compound 3-12

SMILES CNc1ncc(-c2cccc(F)c2)c(N2CC[C@@H]3NCCO[C@H]3C2)c1-c1nc2cc(cc(OC)c2[nH]1)C#N

InChI Key InChIKey=FMTDRTIWTGCPLL-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 527746   

TargetSomatostatin receptor type 2(Human)
Crinetics Pharmaceuticals

US Patent
LigandPNGBDBM527746(US11186590, Compound 3-12)
Affinity DataEC50: >1nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human somatostatin receptor subtype 2 ar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent