BDBM529503 2-(4-fluorophenoxy)-N-::US11203571, Compound 55

SMILES NS(=O)(=O)c1cccc(NC(=O)c2ccc(OC(F)(F)F)cc2Oc2ccc(F)cc2)c1

InChI Key InChIKey=ZUWPJBNZDVNRCL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 529503   

TargetSodium channel protein type 10 subunit alpha(Human)
Vertex Pharmaceuticals

US Patent
LigandPNGBDBM529503(US11203571, Compound 55 | 2-(4-fluorophenoxy)-N-)
Affinity DataIC50: 9nMAssay Description:Patch clamp electrophysiology was used to assess the efficacy and selectivity of sodium channel blockers in dorsal root ganglion neurons. Rat neurons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent