BDBM532032 US11208403, Example 109

SMILES Cc1ccc(cc1)-c1cn(CC2CCOCC2)cc(C(=O)Nc2ccc(nn2)-c2cc(cnc2N)-c2cnn(c2)C2CCOCC2)c1=O

InChI Key InChIKey=GXOVNPXKJGITBD-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 532032   

TargetTyrosine-protein kinase receptor UFO(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM532032(US11208403, Example 109)
Affinity DataIC50: 1.30nMAssay Description:A kinase dilution solution containing 170 ng/ml AXL (the 464th to 885th amino acids of the intracellular domain of human AXL expressed as a fusion pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2022
Entry Details
US Patent

TargetTyrosine-protein kinase Mer(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM532032(US11208403, Example 109)
Affinity DataIC50: 4.00E+3nMAssay Description:A kinase dilution solution containing 20 ng/ml Mer (the 528th to 999th amino acids of the intracellular domain of human MER expressed as a fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2022
Entry Details
US Patent