BDBM577092 5-(4-Chlorophenyl)-7-cyclopropyl-8,9-dihydropyrido[3′,2′: 4,5]pyrrolo[1,2-a]pyrazin-6(7H)-one ::US11472805, Example 9

SMILES Clc1ccc(cc1)-c1c2C(=O)N(CCn2c2ncccc12)C1CC1

InChI Key InChIKey=DVPHOJPLPMGUJK-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 577092   

LigandPNGBDBM577092(US11472805, Example 9 | 5-(4-Chlorophenyl)-7-cyclo...)
Affinity DataIC50: 127nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577092(US11472805, Example 9 | 5-(4-Chlorophenyl)-7-cyclo...)
Affinity DataIC50: 129nMAssay Description:The PDE4A3, PDE4B1, PDE4C1 and PDE4D3 assays use the Scintillation Proximity Assay (SPA) technology to measure the inhibition of human recombinant PD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577092(US11472805, Example 9 | 5-(4-Chlorophenyl)-7-cyclo...)
Affinity DataIC50: 298nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577092(US11472805, Example 9 | 5-(4-Chlorophenyl)-7-cyclo...)
Affinity DataIC50: 8.19E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent