BDBM579449 US11479560, Title ARN-1-770::US11479560, Title ARN-1-776

SMILES CCNC(=O)N1CCC[C@@H](NS(C)(=O)=O)[C@H]1CO[C@H]1CC[C@H](CC1)C(C)C

InChI Key InChIKey=QVBNNVDWURLGGQ-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 579449   

TargetOrexin receptor type 2(Human)
University ff Texas System

US Patent
LigandPNGBDBM579449(US11479560, Title ARN-1-770 | US11479560, Title AR...)
Affinity DataEC50: >500nMAssay Description:HEK293 cells stably expressing OX2R are transfected with Gq alpha construct (6.4 ug per 10 cm dish) using Lipofectamine 3000 (ThermoFisher). 24 hours...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

TargetOrexin receptor type 2(Human)
University ff Texas System

US Patent
LigandPNGBDBM579449(US11479560, Title ARN-1-770 | US11479560, Title AR...)
Affinity DataEC50:  1.50E+3nMAssay Description:HEK293 cells stably expressing OX2R are transfected with Gq alpha construct (6.4 ug per 10 cm dish) using Lipofectamine 3000 (ThermoFisher). 24 hours...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent