BDBM6128 cid_16189061

SMILES CN1C(=O)CCc2cc(-c3cnn(C)c3)c(Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)cc21

InChI Key InChIKey=RPOAJMIQGUOEPW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 6128   

TargetZinc finger and BTB domain-containing protein 7A(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 6128BDBM6128(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (1-met...)
Affinity DataEC50: <10nMAssay Description:Kd values were obtained by incubating His-PPARgamma-LBD with biotinylated peptide, europium-labeled anti-histidine antibody, and allophycocyanin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetProtein Wiz(Homo sapiens)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 6128BDBM6128(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (1-met...)
Affinity DataEC50:  55nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent