BDBM691025 (R)-N-(5-(5-ethylisoxazol-3-yl)-2,3- dihydro-1H-inden-1-yl)-1-methyl-1H- pyrazole-5-carboxamide::US12065436, Compound 414

SMILES CCc1cc(no1)-c1ccc2[C@@H](CCc2c1)NC(=O)c1ccnn1C

InChI Key InChIKey=PUDRGWHTNPDUQC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 691025   

TargetMyosin-1(Bovine)
Cytokinetics

US Patent
LigandPNGBDBM691025((R)-N-(5-(5-ethylisoxazol-3-yl)-2,3- dihydro-1H-in...)
Affinity DataIC50: 600nMAssay Description:To evaluate the effect of compounds on the ATPase activity of full-length cardiac myosin in the context of the native sarcomere, skinned myofibril as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2024
Entry Details
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