BDBM697139 US20240309005, Compound 78

SMILES CN(CCO)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1

InChI Key InChIKey=RFPJRYUBXZJFSL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 697139   

TargetSerine/threonine-protein kinase Sgk1(Human)
Thryv Therapeutics

US Patent
LigandPNGBDBM697139(US20240309005, Compound 78)
Affinity DataIC50: 1.04nMAssay Description:The compounds were tested for SGK-1 activity by measuring the ability of the compound to inhibit the transfer of phosphate from ATP by the isolated e...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/16/2025
Entry Details
US Patent