BDBM71792 2-phenyl-5-(2-piperidin-1-ylethanoylamino)-1,2,3-triazole-4-carboxamide::2-phenyl-5-[(2-piperidin-1-ylacetyl)amino]triazole-4-carboxamide::2-phenyl-5-[(2-piperidinoacetyl)amino]triazole-4-carboxamide::2-phenyl-5-[(piperidin-1-ylacetyl)amino]-2H-1,2,3-triazole-4-carboxamide::5-[[1-oxo-2-(1-piperidinyl)ethyl]amino]-2-phenyl-4-triazolecarboxamide::MLS000045731::SMR000027688::cid_715999
SMILES NC(=O)c1nn(nc1NC(=O)CN1CCCCC1)-c1ccccc1
InChI Key InChIKey=ULZDJPYNTVGZRB-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 71792
TargetIsoform PDE10A2 of cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A (PDE10A2)(Human)
Daiichi Sankyo
US Patent
Daiichi Sankyo
US Patent
Affinity DataIC50: 0.640nMpH: 7.5 T: 2°CAssay Description:A human acute lymphoblastic lymphoma T cell line MOLT-4 (which can be purchased under ATCC No. CRL-1582 from ATCC) was cultured in an RPMI1640 medium...More data for this Ligand-Target Pair
