BDBM722773 US20250059204, Compound 50

SMILES O=S(=O)(Nc3noc4cc(Cn1cccn1)c2CCOc2c34)c5ccccc5OC(F)(F)F

InChI Key InChIKey=SZCBBTBKZJNIQN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 722773   

TargetHistone acetyltransferase KAT6A(Human)
Aurigene Oncology

US Patent
LigandPNGBDBM722773(US20250059204, Compound 50)
Affinity DataIC50: 70nMAssay Description:TR-FRET is homogeneous proximity assay where Europium-labelled anti-acetyl lysine antibody binds to the acetylated substrate labelled with biotin whi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
Go to US Patent