BDBM724674 1-(2-chlorophenyl)-3- methyl-N-((1r,3r)-3- morpholinocyclobut- yl)-1H-thieno[2,3-c] pyrazole-5-carbox- amide::US20250066383, Compound I-3

SMILES Cc1nn(-c2ccccc2Cl)c2sc(C(=O)N[C@H]3C[C@H](N4CCOCC4)C3)cc12

InChI Key InChIKey=HXEGJIXTZSAUKK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 724674   

LigandPNGBDBM724674(1-(2-chlorophenyl)-3- methyl-N-((1r,3r)-3- morphol...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
Go to US Patent

LigandPNGBDBM724674(1-(2-chlorophenyl)-3- methyl-N-((1r,3r)-3- morphol...)
Affinity DataIC50: 65nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
Go to US Patent