BDBM736561 5-((1H-pyrazol-1-yl)methyl)-6-methoxy-N-((5- (trifluoromethyl)-2,3-dihydrobenzofuran-7- yl)sulfonyl)picolinamide::US20250136553, Compound 287

SMILES COc1nc(C(=O)NS(=O)(=O)c2cc(C(F)(F)F)cc3c2OCC3)ccc1Cn1cccn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736561   

TargetHistone acetyltransferase KAT6A(Human)
Olema Pharmaceuticals

US Patent
LigandPNGBDBM736561(5-((1H-pyrazol-1-yl)methyl)-6-methoxy-N-((5- (trif...)
Affinity DataIC50: 11nMAssay Description:TR-FRET based methods were used for assaying compounds of the present invention for KAT6A enzyme inhibitory activity. TR-FRET is a homogeneous proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2025
Entry Details
US Patent