BDBM751716 5-methoxy-2''-(I-methyl-1H-pyrazol-3-yl)-2-morpholino-N-(pyridin-4-yl)-4,4''-bipyrimidin-4-amine ::US20250197375, Compound 56

SMILES COc1c(Nc2ccncc2)nc(N2CCOCC2)nc1-c1ccnc(-c2ccn(C)n2)n1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 751716   

LigandPNGBDBM751716(5-methoxy-2'-(I-methyl-1H-pyrazol-3-yl)-2-morpholi...)
Affinity DataIC50: 550nMAssay Description:Genetic or pharmacological disruption of PIKfyve activity results in enlargement of endosomal vesicles. This enlargement was utilized as a surrogate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent