BDBM764296 US12384777, Example 41

SMILES CCNC(=O)c1cc2c(-c3ccn(C)c(=O)c3Oc3c(C)cc(F)cc3C)cn(C)c(=O)c2[nH]1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 764296   

TargetBromodomain-containing protein 2 [348-455](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: <10nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain-containing protein 4 [348-457](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: <10nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain-containing protein 4 [348-457](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: <10nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain-containing protein 3 [306-416](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: <10nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain testis-specific protein [251-382](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: <10nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: >1.00E+3nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain-containing protein 2 [74-180](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: >3.00E+3nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: >3.00E+3nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain-containing protein 3 [34-140](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: >3.00E+3nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetBromodomain testis-specific protein [27-133](Human)
Tay Therapeutics

US Patent
LigandPNGBDBM764296(US12384777, Example 41)
Affinity DataKd: >3.00E+3nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent