BDBM782783 6''-(((1S,3S)-3-(pyrrolo[2,1-f][1,2,4]triazin-2-ylamino)cyclopentyl)amino)-2H-[1,3''-bipyridinyl]-2-one::US20250326722, Example 20

SMILES O=c1ccccn1c5ccc(N[C@H]4CC[C@H](Nc3ncc2cccn2n3)C4)nc5

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 782783   

TargetProprotein convertase subtilisin/kexin type 9(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM782783(6'-(((1S,3S)-3-(pyrrolo[2,1-f][1,2,4]triazin-2-yla...)
Affinity DataKd:  2.40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/11/2026
Entry Details US Patent