BDBM50038766 3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazole-7-carboxylic acid (3-benzoyl-phenyl)-amide::CHEMBL64449::RP 59227::RP 59228::RP-58467

SMILES O=C(Nc1cccc(c1)C(=O)c1ccccc1)c1ccn2C(SCc12)c1cccnc1

InChI Key InChIKey=PQQFNXGONTVQLM-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50038766   

TargetPlatelet-activating factor receptor(Human)
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50038766(RP 59228 | 3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazol...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50038766(RP 59228 | 3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazol...)
Affinity DataKi:  6.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50038766(RP 59228 | 3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazol...)
Affinity DataKi:  32nMAssay Description:Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50038766(RP 59228 | 3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazol...)
Affinity DataKi:  869nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50038766(RP 59228 | 3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazol...)
Affinity DataKi:  1.36E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details
PubMed