BDBM50011671 (2E,4E)-5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid ((R)-1-methyl-4-pyridin-3-yl-butyl)-amide::5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid (1-methyl-4-pyridin-3-yl-butyl)-amide::CHEMBL277245::Ro-24-0238

SMILES CCCCC\C(=C/C=C/C(=O)N[C@H](C)CCCc1cccnc1)c1ccc(OC)cc1

InChI Key InChIKey=HLCHRSFXEXAMLU-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50011671   

TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011671(CHEMBL277245 | Ro-24-0238 | (2E,4E)-5-(4-Methoxy-p...)
Affinity DataIC50: 40nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011671(CHEMBL277245 | Ro-24-0238 | (2E,4E)-5-(4-Methoxy-p...)
Affinity DataIC50: 40nMAssay Description:Inhibition of [3H]PAF binding to dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011671(CHEMBL277245 | Ro-24-0238 | (2E,4E)-5-(4-Methoxy-p...)
Affinity DataIC50: 40nMAssay Description:Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article