BDBM50071491 4-(1H-Imidazol-4-yl)-butyramidine::CHEMBL72156::SK&F-91606::SK-91606

SMILES NC(=N)CCCc1cnc[nH]1

InChI Key InChIKey=DXLYSPKZUXSVKN-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50071491   

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50071491(4-(1H-Imidazol-4-yl)-butyramidine | SK-91606 | SK&...)
Affinity DataIC50: 1.10nMAssay Description:Histamine H3 receptor agonist activity was assessed by the inhibition of the electrically evoked twitch response of the guinea-pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50071491(4-(1H-Imidazol-4-yl)-butyramidine | SK-91606 | SK&...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of N-alpha-methylhistamine binding to histamine H3 receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed