BDBM85211 t-2,4-PDC::t-PDC

SMILES OC(=O)[C@H]1CN[C@@H](C1)C(O)=O

InChI Key InChIKey=NRSBQSJHFYZIPH-UHFFFAOYSA-N

Data  7 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 85211   

LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for the ability to displace [3H]CGS-19,755 (10 nM) binding in rat forebrain membranes for NMDA receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetExcitatory amino acid transporter 2(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 1(Rat)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetExcitatory amino acid transporter 3(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi:  6.10E+4nMAssay Description:Inhibition of human EAAT3 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetExcitatory amino acid transporter 1(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi:  7.90E+4nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed