BDBM357920 US10214536, Compound 287

SMILES CCOC(=O)c1cc2c(nc1N)Oc3ccc(cc3C2=O)C(C)C

InChI Key InChIKey=PFDJAEKKGJFCNL-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 357920   

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent

LigandBDBM357920(US10214536, Compound 287)Copy SMILESCopy InChI

Affinity DataIC50: 1.23E+5nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchasePC cidPC sidPDBSimilars

In Depth
Date in BDB:
10/20/2019
Entry Details
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PDB3D Structure (crystal)
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