BindingDB BDBM50467836 CHEMBL4282264

BDBM50467836 CHEMBL4282264

SMILES C[C@@H](C(F)(F)F)N(Cc1ccc(cc1)F)C(=O)CN2C(=O)[C@]3(CCc4c3ccc(c4)NC(=O)NC)OC2=O

InChI Key InChIKey=VRVJKILQRBSEAG-UHFFFAOYSA-N

Data 94 IC50 3 Kd 3 EC50

PDB links: 1 PDB ID matches this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 100 hits for monomerid = 50467836

Tyrosine-protein kinase Lck(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Platelet-derived growth factor receptor beta(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Platelet-derived growth factor receptor alpha(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase PAK 4(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

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Date in BDB:
10/13/2025
Entry Details
PubMed

Mitogen-activated protein kinase 14(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase Nek2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase 4(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

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Date in BDB:
10/13/2025
Entry Details
PubMed

Dual specificity mitogen-activated protein kinase kinase 2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Dual specificity mitogen-activated protein kinase kinase 1(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Mitogen-activated protein kinase kinase kinase kinase 4(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Mitogen-activated protein kinase kinase kinase kinase 2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
GoogleScholar

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Date in BDB:
10/13/2025
Entry Details
PubMed

Mitogen-activated protein kinase kinase kinase 10(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Dual specificity mitogen-activated protein kinase kinase 3(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

cAMP-dependent protein kinase catalytic subunit gamma(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
GoogleScholar

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Date in BDB:
10/13/2025
Entry Details
PubMed

Leukocyte tyrosine kinase receptor(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Vascular endothelial growth factor receptor 2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Mitogen-activated protein kinase 9(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Mitogen-activated protein kinase 8(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Tyrosine-protein kinase JAK3(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Tyrosine-protein kinase JAK2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Insulin receptor(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Inhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Insulin-like growth factor 1 receptor(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Glycogen synthase kinase-3 beta(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
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Date in BDB:
10/13/2025
Entry Details
PubMed

Glycogen synthase kinase-3 alpha(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase 16(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Death-associated protein kinase 3(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Wee1-like protein kinase(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

NT-3 growth factor receptor(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

BDNF/NT-3 growth factors receptor(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

High affinity nerve growth factor receptor(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Tyrosine-protein kinase receptor TYRO3(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Activated CDC42 kinase 1(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase TBK1(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase TAO2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Tyrosine-protein kinase SYK(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Proto-oncogene tyrosine-protein kinase Src(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase 33(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

G protein-coupled receptor kinase 5(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase Sgk1(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Ribosomal protein S6 kinase alpha-3(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Rho-associated protein kinase 2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Rho-associated protein kinase 1(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Proto-oncogene tyrosine-protein kinase receptor Ret(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase D3(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase pim-2(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Serine/threonine-protein kinase pim-1(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

cGMP-dependent protein kinase 1(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Protein kinase C zeta type(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Date in BDB:
10/13/2025
Entry Details
PubMed

Protein kinase C theta type(Human)
AbbVie

Curated by ChEMBL

PNG

BDBM50467836(CHEMBL4282264)

IC50: 1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

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Date in BDB:
10/13/2025
Entry Details
PubMed

Displayed 1 to 50 (of 100 total ) | Next | Last >>

Filter my 100 hits

Targets 81▿
- Histone acetyltransferase p300 15
- CREB-binding protein 4
- Platelet-derived growth factor receptor alpha/beta 3
- Serine/threonine-protein kinase D3 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1B 1
- Death-associated protein kinase 3 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 1
- Serine/threonine-protein kinase pim-1 1
- Serine/threonine-protein kinase pim-2 1
- Cyclin-dependent kinase 11B 1
- Calcium/calmodulin-dependent protein kinase kinase 2 1
- Serine/threonine-protein kinase TAO2 1
- Mitogen-activated protein kinase kinase kinase kinase 2 1
- Mitogen-activated protein kinase kinase kinase kinase 4 1
- ALK tyrosine kinase receptor 1
- Hepatocyte growth factor receptor 1
- Mitogen-activated protein kinase 14 1
- Serine/threonine-protein kinase B-raf 1
- Glycogen synthase kinase-3 alpha 1
- Leukocyte tyrosine kinase receptor 1
- Glycogen synthase kinase-3 beta 1
- Bromodomain-containing protein 4 1
- Bromodomain-containing protein 3 1
- Serine/threonine-protein kinase Nek2 1
- Tyrosine-protein kinase ABL1 1
- Protein kinase C theta type 1
- RAC-alpha serine/threonine-protein kinase 1
- Dual specificity mitogen-activated protein kinase kinase 2 1
- Serine/threonine-protein kinase PAK 4 1
- Dual specificity mitogen-activated protein kinase kinase 3 1
- Calcium/calmodulin-dependent protein kinase type II subunit alpha 1
- Tyrosine-protein kinase JAK3 1
- Dual specificity mitogen-activated protein kinase kinase 1 1
- Tyrosine-protein kinase JAK2 1
- Proto-oncogene tyrosine-protein kinase receptor Ret 1
- cGMP-dependent protein kinase 1 1
- Rho-associated protein kinase 2 1
- Bromodomain testis-specific protein 1
- Rho-associated protein kinase 1 1
- Serine/threonine-protein kinase Sgk1 1
- Proto-oncogene tyrosine-protein kinase Src 1
- BDNF/NT-3 growth factors receptor 1
- Mitogen-activated protein kinase 1 1
- Tyrosine-protein kinase Lck 1
- Serine/threonine-protein kinase 4 1
- Tyrosine-protein kinase BTK 1
- NT-3 growth factor receptor 1
- Mitogen-activated protein kinase 9 1
- G protein-coupled receptor kinase 5 1
- Insulin-like growth factor 1 receptor 1
- Dual specificity protein kinase CLK2 1
- High affinity nerve growth factor receptor 1
- Serine/threonine-protein kinase 16 1
- Epidermal growth factor receptor 1
- Mitogen-activated protein kinase 8 1
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
- Tyrosine-protein kinase SYK 1
- Ribosomal protein S6 kinase alpha-3 1
- Serine/threonine-protein kinase TBK1 1
- Calcium/calmodulin-dependent protein kinase type 1D 1
- Aurora kinase B 1
- Insulin receptor 1
- Vascular endothelial growth factor receptor 2 1
- Fibroblast growth factor receptor 1 1
- Aurora kinase A 1
- Vascular endothelial growth factor receptor 1 1
- Wee1-like protein kinase 1
- Serine/threonine-protein kinase PLK3 1
- Tyrosine-protein kinase receptor TYRO3 1
- Casein kinase I isoform alpha 1
- Tyrosine-protein kinase Fyn 1
- Macrophage colony-stimulating factor 1 receptor 1
- Focal adhesion kinase 1 1
- Platelet-derived growth factor receptor alpha 1
- Protein kinase C zeta type 1
- Serine/threonine-protein kinase 33 1
- cAMP-dependent protein kinase catalytic subunit gamma 1
- Activated CDC42 kinase 1 1
- Platelet-derived growth factor receptor beta 1
- Epithelial discoidin domain-containing receptor 1 1
- Mitogen-activated protein kinase kinase kinase 10 1
Publications 11▿
- Nature 550: 128-132 85
- ACS Med Chem Lett 12: 726-731 (2021) 2
- J Med Chem 67: 5351-5372 2
- Bioorg Med Chem 52: (2021) 2
- J Med Chem 63: 1337-1360 (2020) 2
- J Med Chem 67: 5275-5304 2
- Bioorg Med Chem 26: 5397-5407 (2018) 1
- Eur J Med Chem 266: 1
- Eur J Med Chem 237: (2022) 1
- J Med Chem 63: 4716-4731 (2020) 1
- J Med Chem 62: 7146-7159 (2019) 1
Institutions 9▿
- AbbVie 85
- University of Michigan 4
- Chinese Academy of Sciences 3
- China Pharmaceutical University 2
- Abbvie 2
- Baylor College of Medicine 1
- Sichuan University 1
- Cancer Therapeutics Crc 1
- Avera Institute For Human Genetics 1
Affinity: 0.0013 to 1.0E+4 nM▿
- IC50 94
- Kd 3
- EC50 3
- Affinity ≤ nM
Xtal structures: 1
Docked structures: 0
Catalog Cmpds: 1