Compile Data Set for Download or QSAR
Report error Found 23030 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2'
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKd:  0.220nMAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKd:  0.220nMpH: 7.4 T: 2°CAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKd:  0.330nMAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21222(N-[6-methoxy-2-(methylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21223(N-[6-methoxy-2-(methylsulfanyl)pyrimidin-4-yl]prop...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21226(N-[6-methoxy-2-(propylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21227(N-[6-methoxy-2-(propylsulfanyl)pyrimidin-4-yl]prop...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21228(N-[6-propoxy-2-(propylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21230(N-[2-(benzylsulfanyl)-6-propoxypyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21231(N-[6-(benzyloxy)-2-(propylsulfanyl)pyrimidin-4-yl]...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21233(N-{6-[(3-chlorophenyl)methoxy]-2-(propylsulfanyl)p...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21234(N-{6-[(4-chlorophenyl)methoxy]-2-(propylsulfanyl)p...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21235(N-{6-[(2,4-dichlorophenyl)methoxy]-2-(propylsulfan...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21236(N-{6-[(4-methoxyphenyl)methoxy]-2-(propylsulfanyl)...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21237(N-[6-(2-phenylethoxy)-2-(propylsulfanyl)pyrimidin-...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21238(N-[6-(cyclohexylmethoxy)-2-(propylsulfanyl)pyrimid...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21239(N-{6-[(4-chlorophenyl)methoxy]-2-(ethylsulfanyl)py...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM21240(N-[2-(tert-butylsulfanyl)-6-[(4-chlorophenyl)metho...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  140nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59202(Adenosine analog, 5)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM50208817(CHEMBL376542 | Adenosine analog, 6 | (2S,3S,4R,5R)...)
Affinity DataEC50:  54.5nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM50185934(CHEMBL378606 | Adenosine analog, 7 | (2S,3S,4R,5R)...)
Affinity DataEC50:  1.20E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM50106539(5'-N-[(2-AMINO)ETHYL CARBOXAMIDO] ADENOSINE | 5-(6...)
Affinity DataEC50:  1.56E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59203(Adenosine analog, 8)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59204(Adenosine analog, 9)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59205(Adenosine analog, 10)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59206(Adenosine analog, 11)
Affinity DataEC50:  942nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59207(Adenosine analog, 12)
Affinity DataEC50: >1.00E+5nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59208(Adenosine analog, 13)
Affinity DataEC50: >1.00E+3nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59209(Adenosine analog, 14)
Affinity DataEC50: >1.00E+3nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59210(Adenosine analog, 15)
Affinity DataEC50:  3.72E+3nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM50163021(Adenosine analog, 17 | CHEMBL194830 | (2R,3R,4S,5R...)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59211(Adenosine analog, 18)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
National Institutes of Health

LigandPNGBDBM59212(Adenosine analog, 19)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2011
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191774(US9187428, 2)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191775(US9187428, 3)
Affinity DataEC50:  425nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191776(US9187428, 53 | US9187428, 4)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191778(US9187428, 6)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191779(US9187428, 7)
Affinity DataEC50:  460nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191785(US9187428, 13)
Affinity DataEC50:  108nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191786(US9187428, 14)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191787(US9187428, 15)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191793(US9187428, 21)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191798(US9187428, 26)
Affinity DataEC50:  65nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191799(US9187428, 27)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191800(US9187428, 28)
Affinity DataEC50:  1.64E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191801(US9187428, 29)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191802(US9187428, 30)
Affinity DataEC50:  1.11E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191803(US9187428, 31)
Affinity DataEC50:  707nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Neuroscience

LigandPNGBDBM191804(US9187428, 32)
Affinity DataEC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

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