Report error Found 2570 Enz. Inhib. hit(s) with Target = 'Amyloid-beta precursor protein'
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Inhibitory activity against binding of [125I]IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Inhibitory activity against binding of [125I]IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Inhibitory activity against binding of [125I]IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Inhibition constant for aggregates of amyloid beta compared to [125I]-IMSBMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Inhibitory activity against binding of [125I]IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]PIB from amyloid beta (1 to 42) aggregates in Alzheimer's disease-human brain homogenate after 3 hrs by gamma countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.208nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKd: 0.210nMAssay Description:Displacement of [125I-N-Methyl-4-(4-bromoanilino)phthalimide from beta-amyloid plaques isolated from Alzheimer's disease patient brainMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Inhibitory activity against binding of [125I]IMSB to amyloid beta in brainMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of gamma-secretase assessed as reduction of membrane A-beta-40 levelMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]PIB from amyloid beta (1 to 42) aggregates in Alzheimer's disease-human brain homogenate after 3 hrs by gamma countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.380nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition constant of compound on ligand binding to aggregates of Amyloid beta was measured by comparing with [125I]-IMSBMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.560nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.560nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKd: 0.560nMAssay Description:Binding affinity to amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.590nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.600nMT: 2°CAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at -140 C. at a concent...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.620nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:The β-secretase enzyme used in the TR-FRET is prepared as follows: The cDNA for the soluble part of the human β-Secretase (AA 1-AA 460) was...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.700nMT: 2°CAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at -140 C. at a concent...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:The β-secretase enzyme used in the TR-FRET is prepared as follows: The cDNA for the soluble part of the human β-Secretase (AA 1-AA 460) was...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:The β-secretase enzyme used in the TR-FRET is prepared as follows: The cDNA for the soluble part of the human β-Secretase (AA 1-AA 460) was...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.700nMT: 2°CAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at -140 C. at a concent...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [125I]IMPY from beta amyloid in human corpse AD brainMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:The β-secretase enzyme used in the TR-FRET is prepared as follows: The cDNA for the soluble part of the human β-Secretase (AA 1-AA 460) was...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [18F]-amyvid from amyloid-beta aggregates in alzheimer's disease patient brain homogenates after 1 hrMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Binding affinity to Beta amyloid aggregates in Alzheimer's disease patient brain by competitive binding assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.780nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Sungkyunkwan University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:SH-SY5Y cells were cultured in DMEM/F-12 with Glutamax, 10% FCS and 1% non-essential amino acids and cryopreserved and stored at −140° C. at a ...More data for this Ligand-Target Pair

































