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Report error Found 38 Enz. Inhib. hit(s) with Target = 'C-C motif chemokine 5'
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017345(CHEMBL3288260)
Affinity DataKd:  2.50E+7nMAssay Description:Binding affinity to human recombinant CCL5 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017347(CHEMBL3288259)
Affinity DataKd:  2.50E+7nMAssay Description:Binding affinity to human recombinant CCL5 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017346(CHEMBL3288258)
Affinity DataKd:  2.50E+7nMAssay Description:Binding affinity to human recombinant CCL5 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50585055(CHEMBL5081237)
Affinity DataKd:  5.72E+3nMAssay Description:Binding affinity to human CCL5 assessed as dissociation constant incubated for 3 mins by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329229((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-phenyl...)
Affinity DataIC50: 17nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329246(((3aR,6aS)-5-(3-(1-(cyclopentylsulfonyl)azetidin-3...)
Affinity DataIC50: 22nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329250(((3aR,6aS)-5-(3-(1-(cyclopentylsulfonyl)piperidin-...)
Affinity DataIC50: 23nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329241((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(1-(is...)
Affinity DataIC50: 23nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329249((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(1-(et...)
Affinity DataIC50: 25nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329232(((3aR,6aS)-5-(3-(1-(2,2-difluoroethyl)piperidin-4-...)
Affinity DataIC50: 25nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329230(((3aR,6aS)-5-(3-(1-(2,2-difluoroethyl)piperidin-4-...)
Affinity DataIC50: 27nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329248(((3aR,6aS)-5-(3-(1-(cyclopropylsulfonyl)piperidin-...)
Affinity DataIC50: 27nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329255(4,6-dimethyl-5-((3aR,6aS)-5-(3-(1-(methylsulfonyl)...)
Affinity DataIC50: 27nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329256(4,6-dimethyl-5-((3aR,6aS)-5-(3-(1-(methylsulfonyl)...)
Affinity DataIC50: 31nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329235(1-(4-(3-((3aR,6aS)-5-(4,6-dimethylpyrimidine-5-car...)
Affinity DataIC50: 32nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329251((4,6-dimethyl pyrimidin-5-yl)((3aR,6aS)-5-(3-(1-(m...)
Affinity DataIC50: 34nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329251((4,6-dimethyl pyrimidin-5-yl)((3aR,6aS)-5-(3-(1-(m...)
Affinity DataIC50: 34nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329244(((3aR,6aS)-5-(3-(1-(cyclopropylsulfonyl)azetidin-3...)
Affinity DataIC50: 35nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329231(((3aR,6aS)-5-(3-(1-(2,2-difluoroethyl)piperidin-4-...)
Affinity DataIC50: 35nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329252((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(3-flu...)
Affinity DataIC50: 38nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329243(((3aR,6aS)-5-(3-(1-(cyclopropylsulfonyl)azetidin-3...)
Affinity DataIC50: 39nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329242(((3aR,6aS)-5-(3-(1-(cyclopropylsulfonyl)azetidin-3...)
Affinity DataIC50: 40nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329227((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(3-flu...)
Affinity DataIC50: 44nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329227((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(3-flu...)
Affinity DataIC50: 44nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329234((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(1-(is...)
Affinity DataIC50: 47nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329247((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-phenyl...)
Affinity DataIC50: 48nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329245((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(1-(me...)
Affinity DataIC50: 52nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329237(1-(4-(3-((3aR,6aS)-5-(4,6-dimethylpyrimidine-5-car...)
Affinity DataIC50: 68nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329236(1-(4-(3-((3aR,6aS)-5-(4,6-dimethylpyrimidine-5-car...)
Affinity DataIC50: 72nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329233(methyl 4-(3-((3aR,6aS)-5-(4,6-dimethylpyrimidine-5...)
Affinity DataIC50: 102nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329253((2-chloro-6-methylphenylsulfonyl)((3aR,6aS)-5-(3-(...)
Affinity DataIC50: 104nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329239(((3aR,6aS)-5-(3-(1-(cyclopentanecarbonyl)azetidin-...)
Affinity DataIC50: 207nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329254(3-chloro-4-((3aR,6aS)-5-(3-(1-(methylsulfonyl)pipe...)
Affinity DataIC50: 215nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329240(1-(3-(3-((3aR,6aS)-5-(4,6-dimethylpyrimidine-5-car...)
Affinity DataIC50: 500nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329238((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-phenyl...)
Affinity DataIC50: 500nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329251((4,6-dimethyl pyrimidin-5-yl)((3aR,6aS)-5-(3-(1-(m...)
Affinity DataIC50: 500nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329227((4,6-dimethylpyrimidin-5-yl)((3aR,6aS)-5-(3-(3-flu...)
Affinity DataIC50: 500nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetC-C motif chemokine 5(Human)
Momenta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50329228(4-(3-((3aR,6aS)-5-(4,6-dimethylpyrimidine-5-carbon...)
Affinity DataIC50: 500nMAssay Description:Inhibition of RANTESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed