Compile Data Set for Download or QSAR
Report error Found 266 Enz. Inhib. hit(s) with Target = 'Choline kinase'
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145944(CHEMBL3763540)
Affinity DataKd:  10nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579779(CHEMBL5091519)
Affinity DataIC50: 14nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579781(CHEMBL5094847)
Affinity DataIC50: 14nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50146014(CHEMBL3765554)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human ChoKalpha using choline as substrate by ultraviolet spectroscopic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579773(CHEMBL5079663)
Affinity DataIC50: 20nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579782(CHEMBL5078600)
Affinity DataIC50: 20nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579777(CHEMBL5090932)
Affinity DataIC50: 21nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145945(CHEMBL3764278)
Affinity DataKd:  21nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579771(CHEMBL5077194)
Affinity DataIC50: 22nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579769(CHEMBL5075042)
Affinity DataIC50: 23nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579780(CHEMBL5089356)
Affinity DataIC50: 27nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579757(CHEMBL5084844)
Affinity DataIC50: 28nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579775(CHEMBL5085262)
Affinity DataIC50: 28nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579770(CHEMBL5090132)
Affinity DataIC50: 29nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579774(CHEMBL5081222)
Affinity DataIC50: 31nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579785(CHEMBL5075110)
Affinity DataIC50: 31nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579786(CHEMBL5093152)
Affinity DataIC50: 31nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579772(CHEMBL5088776)
Affinity DataIC50: 33nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579784(CHEMBL5091201)
Affinity DataIC50: 34nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579764(CHEMBL5086885)
Affinity DataIC50: 40nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579778(CHEMBL5078057)
Affinity DataIC50: 43nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579758(CHEMBL5085127)
Affinity DataIC50: 49nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579783(CHEMBL5088850)
Affinity DataIC50: 49nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579765(CHEMBL5089748)
Affinity DataIC50: 61nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145944(CHEMBL3763540)
Affinity DataIC50: 66nMAssay Description:Inhibition of human N-terminal truncated ChoKalpha1 (75 to 457 residues) using choline chloride as substrate measured over 10 to 30 mins by coupled A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145946(CHEMBL3763931)
Affinity DataIC50: 85nMAssay Description:Inhibition of human N-terminal truncated ChoKalpha1 (75 to 457 residues) using choline chloride as substrate measured over 10 to 30 mins by coupled A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579766(CHEMBL5093251)
Affinity DataIC50: 88nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145947(CHEMBL3763792)
Affinity DataKd:  88nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579776(CHEMBL5077317)
Affinity DataIC50: 97nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145946(CHEMBL3763931)
Affinity DataKd:  99nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579767(CHEMBL5089440)
Affinity DataIC50: 104nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50447102(CHEMBL3112879)
Affinity DataKd:  110nMAssay Description:Binding affinity to human CK-alpha1 by tryptophan fluorescence spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579759(CHEMBL5075746)
Affinity DataIC50: 111nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579760(CHEMBL5085340)
Affinity DataIC50: 126nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579761(CHEMBL5087533)
Affinity DataIC50: 138nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579768(CHEMBL5094938)
Affinity DataIC50: 146nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579762(CHEMBL5086986)
Affinity DataIC50: 151nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145989(CHEMBL3763982)
Affinity DataIC50: 165nMAssay Description:Inhibition of human N-terminal truncated ChoKalpha1 (75 to 457 residues) using choline chloride as substrate measured over 10 to 30 mins by coupled A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50556492(CHEMBL4747352)
Affinity DataKd:  185nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145942(CHEMBL3765239)
Affinity DataKd:  195nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145989(CHEMBL3763982)
Affinity DataKd:  211nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579741(CHEMBL5076272)
Affinity DataIC50: 227nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145945(CHEMBL3764278)
Affinity DataIC50: 233nMAssay Description:Inhibition of human N-terminal truncated ChoKalpha1 (75 to 457 residues) using choline chloride as substrate measured over 10 to 30 mins by coupled A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579729(CHEMBL5092659)
Affinity DataIC50: 236nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579734(CHEMBL5091650)
Affinity DataIC50: 248nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579742(CHEMBL5094399)
Affinity DataIC50: 249nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145942(CHEMBL3765239)
Affinity DataIC50: 251nMAssay Description:Inhibition of human N-terminal truncated ChoKalpha1 (75 to 457 residues) using choline chloride as substrate measured over 10 to 30 mins by coupled A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50146003(CHEMBL3763453)
Affinity DataIC50: 255nMAssay Description:Inhibition of human N-terminal truncated ChoKalpha1 (75 to 457 residues) using choline chloride as substrate measured over 10 to 30 mins by coupled A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50146003(CHEMBL3763453)
Affinity DataKd:  259nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145947(CHEMBL3763792)
Affinity DataIC50: 268nMAssay Description:Inhibition of human N-terminal truncated ChoKalpha1 (75 to 457 residues) using choline chloride as substrate measured over 10 to 30 mins by coupled A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
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