Compile Data Set for Download or QSAR
Report error Found 656 Enz. Inhib. hit(s) with Target = 'Endoplasmin'
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210939(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-phenyl...)
Affinity DataKd:  9.05E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210940(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(o-tol...)
Affinity DataKd:  9.90E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210941(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(m-tol...)
Affinity DataKd:  9.43E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210942(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(p-tol...)
Affinity DataKd:  8.35E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210943(4-(2-(2-chlorophenyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  2.94E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210944(4-(2-(3-chlorophenyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  1.58E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210945(4-(2-(4-chlorophenyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  1.06E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210946(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(pyrid...)
Affinity DataKd:  1.40E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210947(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(pyrid...)
Affinity DataKd:  5.50E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210948(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(pyrid...)
Affinity DataKd:  1.32E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210949(4-(2-benzyl-1H-pyrrol-1-yl)-2-(((1r,4r)-4-hydroxyc...)
Affinity DataKd:  1.13E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210950(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-phenet...)
Affinity DataKd: >2.50E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210951(4-(2-(2-chlorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  830nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210952(4-(2-(3-chlorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  2.45E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210953(4-(2-(4-chlorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd: >2.50E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210954(4-(2-(2-fluorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  720nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210955(4-(2-(3-fluorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  4.53E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210956(4-(2-(4-fluorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  8.35E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210957(4-(2-(2-bromobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-4...)
Affinity DataKd:  1.29E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210958(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(2-met...)
Affinity DataKd:  4.20E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210959(4-(2-(2-hydroxybenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)...)
Affinity DataKd:  440nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210960(4-(2-(3-hydroxybenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)...)
Affinity DataKd: >2.50E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210961(4-(2-(4-hydroxybenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)...)
Affinity DataKd:  2.06E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210962(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(2-met...)
Affinity DataKd:  1.15E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210963(4-(2-(2,6-difluorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,...)
Affinity DataKd: >2.50E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210964(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(pyrid...)
Affinity DataKd:  1.40E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210965(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(pyrid...)
Affinity DataKd:  5.50E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
The University of Kansas

LigandPNGBDBM210966(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(pyrid...)
Affinity DataKd:  1.32E+4nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501623(US11028041, Compound 6)
Affinity DataKd:  630nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501624(US11028041, Compound 7)
Affinity DataKd:  1.04E+4nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501625(US11028041, Compound 16)
Affinity DataKd:  450nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501626(US11028041, Compound 17)
Affinity DataKd:  680nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501627(US11028041, Compound 18)
Affinity DataKd:  730nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501628(US11028041, Compound 19)
Affinity DataKd:  280nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501629(US11028041, Compound 20)
Affinity DataKd:  240nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501630(US11028041, Compound 21)
Affinity DataKd:  180nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501631(US11028041, Compound 22)
Affinity DataKd:  300nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501632(US11028041, Compound 23)
Affinity DataKd:  330nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501633(US11028041, Compound 24)
Affinity DataKd:  540nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501634(US11028041, Compound 25)
Affinity DataKd:  6.10E+3nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501635(US11028041, Compound 26)
Affinity DataKd:  7.80E+3nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501636(US11028041, Compound 27)
Affinity DataKd:  5.50E+3nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501637(US11028041, Compound 28)
Affinity DataKd:  1.19E+4nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501638(US11028041, Compound 29)
Affinity DataKd:  4.20E+3nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM50450703(CHEMBL4159086 | US11028041, Compound 30)
Affinity DataKd:  540nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM501640(US11028041, Compound 31)
Affinity DataKd:  360nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
US Patent

TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM50279156(CHEMBL4169566)
Affinity DataKd:  31nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM50279157(CHEMBL4168916)
Affinity DataKd:  9.89E+3nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM50279158(CHEMBL4175693)
Affinity DataKd:  34nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
University of Kansas

US Patent
LigandPNGBDBM50279170(CHEMBL4162283)
Affinity DataKd:  59nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
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