Compile Data Set for Download or QSAR
Report error Found 217 Enz. Inhib. hit(s) with Target = 'Enoyl-acyl-carrier protein reductase'
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  0.00190nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGCG by dilution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  0.0521nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of ECG by dilution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  0.109nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGC by dilution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  0.281nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of quercetin by dilution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  0.798nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of butein by dilution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  1nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGCGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50211885(5-(3,4-dihydroxybenzylidene)-3-phenyl-2-thioxothia...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of Plasmodium falciparum recombinant enoyl ACP reductase expressed in BL21 (DE3) cells with respect to crotonyl CoAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  7.29nMAssay Description:Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of EGCGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  8nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of ECGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataKi:  8nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  8.25nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  10nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of quercetinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  13.7nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of buteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50042949((E)-3-(3,4-Dihydroxy-phenyl)-1-(2,4-dihydroxy-phen...)
Affinity DataKi:  14nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50153015((-)epicatechingallate | (2R,3R)-2-(3,4-dihydroxyph...)
Affinity DataKi:  16nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50187665((-)-epigallocatechin | CHEMBL47386)
Affinity DataKi:  17.6nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataKi:  22nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  28.3nMAssay Description:Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of ECGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  30.5nMAssay Description:Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of quercetinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50211885(5-(3,4-dihydroxybenzylidene)-3-phenyl-2-thioxothia...)
Affinity DataKi:  32nMAssay Description:Inhibition of Plasmodium falciparum recombinant enoyl ACP reductase expressed in BL21 (DE3) cells with respect to NADHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50211885(5-(3,4-dihydroxybenzylidene)-3-phenyl-2-thioxothia...)
Affinity DataIC50: 35nMAssay Description:Inhibition of Plasmodium falciparum recombinant enoyl ACP reductase expressed in BL21 (DE3) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50135169((2S,3R)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-3,4-...)
Affinity DataKi:  40nMAssay Description:Inhibition of FabIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  50nMAssay Description:Inhibition of Plasmodium falciparum enoyl-acyl carrier protein reductase expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  52.7nMAssay Description:Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of EGCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174772(N-(3-chloro-4-(4-chloro-2-hydroxyphenoxy)phenyl)ac...)
Affinity DataIC50: 57nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataIC50: 66nMAssay Description:Inhibition of Plasmodium falciparum recombinant enoyl ACP reductase expressed in BL21 (DE3) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataIC50: 70nMAssay Description:Inhibition of Plasmodium falciparum recombinant FabIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataIC50: 70nMAssay Description:Inhibition of Plasmodium falciparum enoyl-ACP reductase assessed as oxidation of NADH to NAD+ after 10 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM25419(5-benzyl-2-(2,4-dichlorophenoxy)phenol | Triclosan...)
Affinity DataIC50: 71nMAssay Description:Inhibition of Plasmodium falciparum enoyl-acyl carrier protein reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataKi:  71.0nMAssay Description:Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of buteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataIC50: 73nMAssay Description:Inhibition of Plasmodium falciparum ENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataIC50: 73nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM8726(CHEMBL849 | TCL | 5-chloro-2-(2,4-dichlorophenoxy)...)
Affinity DataIC50: 73nMAssay Description:Inhibition of Plasmodium falciparum enoyl-acyl carrier protein reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM25420(2-(2,4-dichlorophenoxy)-5-(2-phenylethyl)phenol | ...)
Affinity DataIC50: 76nMAssay Description:Inhibition of Plasmodium falciparum enoyl-acyl carrier protein reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataKi:  79nMAssay Description:Inhibition of Plasmodium falciparum ENR using crotonyl-CoA substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50153015((-)epicatechingallate | (2R,3R)-2-(3,4-dihydroxyph...)
Affinity DataKi:  102nMAssay Description:Inhibition of Plasmodium falciparum ENR using crotonyl-CoA substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM25412(2-(2,4-dichlorophenoxy)-5-(3-methylbutyl)phenol | ...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Plasmodium falciparum enoyl-acyl carrier protein reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174775(3-chloro-4-(4-chloro-2-hydroxyphenoxy)benzonitrile...)
Affinity DataIC50: 120nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174766(3-chloro-4-(4-chloro-2-hydroxyphenoxy)benzamide | ...)
Affinity DataIC50: 120nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174769(N-(3-chloro-4-(4-chloro-2-hydroxyphenoxy)phenyl)tr...)
Affinity DataIC50: 140nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174760(CHEMBL200585 | 2‐[4‐(benzylamino)̴...)
Affinity DataIC50: 140nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174778(1-(3-chloro-4-(4-chloro-2-hydroxyphenoxy)phenyl)ur...)
Affinity DataIC50: 160nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174776(N-(3-chloro-4-(4-chloro-2-hydroxyphenoxy)phenyl)be...)
Affinity DataIC50: 170nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM25410(2-(2,4-dichlorophenoxy)-5-(2-methylpropyl)phenol |...)
Affinity DataIC50: 180nMAssay Description:Inhibition of Plasmodium falciparum enoyl-acyl carrier protein reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174770(5-chloro-2-(2-chloro-4-nitrophenoxy)phenol | CHEMB...)
Affinity DataIC50: 180nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataKi:  186nMAssay Description:Inhibition of Plasmodium falciparum ENR using NADH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174767(2-(3-chloro-4-(4-chloro-2-hydroxyphenoxy)phenyl)ac...)
Affinity DataIC50: 190nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM25417(2-(2,4-dichlorophenoxy)-5-(4-methylphenyl)phenol |...)
Affinity DataIC50: 190nMAssay Description:Inhibition of Plasmodium falciparum enoyl-acyl carrier protein reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50174754((3-chloro-4-(4-chloro-2-hydroxyphenoxy)phenyl)(mor...)
Affinity DataIC50: 200nMAssay Description:Inhibition of PfENR enzymatic activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEnoyl-acyl-carrier protein reductase(malaria parasite P. falciparum)
National Institute of Immunology

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataIC50: 200nMAssay Description:Inhibition of FabIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
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