Report error Found 875 Enz. Inhib. hit(s) with Target = 'Fatty acid-binding protein, adipocyte'
Displayed 1 to 50 (of 875 total ) | Next | Last >>
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Binding affinity to FABP4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: <2nMAssay Description:Inhibition of human FABP4 assessed as inhibition constant by fluorescent displacement assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to ap2More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKd: 4nMAssay Description:Binding affinity to human FABP4 expressed in Escherichia coli assessed as degree of fluorescent shift by temperature-dependent fluorescence thermal s...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of fluorescent 1-anilinonapthalene 8-sulfonic acid from human a-FABP by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of fluorescent 1-anilinonapthalene 8-sulfonic acid from human a-FABP by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of fluorescent 1-anilinonapthalene 8-sulfonic acid from human a-FABP by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of Bodipy-labeled fatty acid from recombinant human His6-tagged FABP4 expressed in Escherichia coli after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to recombinant FABP4 (unknown origin) expressed in Escherichia coli by sypro orange dye-based TdF assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human FABP4More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human FABP4More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to human FABP4 expressed in Escherichia coli assessed as degree of fluorescent shift by temperature-dependent fluorescence thermal s...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 11nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of Bodipy-labeled fatty acid from recombinant human His6-tagged FABP4 expressed in Escherichia coli after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of FABP4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of Bodipy-labeled fatty acid from recombinant human His6-tagged FABP4 expressed in Escherichia coli after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 13nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of Bodipy-labeled fatty acid from recombinant human His6-tagged FABP4 expressed in Escherichia coli after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of fluorescent 1-anilinonapthalene 8-sulfonic acid from human a-FABP by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Human)
Universita degli Studi di Catania
Curated by ChEMBL
Universita degli Studi di Catania
Curated by ChEMBL
Affinity DataIC50: 13nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair














































