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Report error Found 342 Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 1'
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataEC50:  0.0614nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | TCMDC-12...)
Affinity DataEC50:  1.49nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM73209(cid_657346 | methamilane methiodide | trimethyl-[[...)
Affinity DataEC50:  0.280nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM34572(UK 14,304 | SMR000058355 | CHEMBL844 | cid_2435 | ...)
Affinity DataEC50:  0.0372nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM73210(SMR000030412 | MLS000094859 | (5Z)-5-{(2E)-3-[4-(d...)
Affinity DataEC50:  0.856nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM36882(3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5,7-dihydroxy...)
Affinity DataEC50:  1.26E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM42613(cid_657947 | SMR000059240 | 3-prop-2-enyl-2-sulfan...)
Affinity DataEC50:  3.15E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM73211(1-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[1,1,1...)
Affinity DataEC50:  2.29E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM73212(cid_2955604 | SMR000076705 | ethyl 4-[({[1-(tetrah...)
Affinity DataEC50:  4.14E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497366(CHEMBL3339138)
Affinity DataEC50:  4.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497367(CHEMBL3339146)
Affinity DataEC50:  310nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497368(CHEMBL3339126)
Affinity DataEC50:  3.00E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497375(CHEMBL3339133)
Affinity DataEC50:  990nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497382(CHEMBL3339124)
Affinity DataEC50:  1.30E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497383(CHEMBL3339129)
Affinity DataEC50:  660nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497384(CHEMBL3339128)
Affinity DataEC50:  270nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497374(CHEMBL3339127)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497385(CHEMBL3339123)
Affinity DataEC50:  890nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497379(CHEMBL3339121)
Affinity DataEC50:  460nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497386(CHEMBL3339132)
Affinity DataEC50:  520nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497376(CHEMBL3339134)
Affinity DataEC50:  780nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497387(CHEMBL3339135)
Affinity DataEC50:  780nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497388(CHEMBL3339137)
Affinity DataEC50:  730nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497389(CHEMBL3339139)
Affinity DataEC50:  3.80E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497380(CHEMBL3339140)
Affinity DataEC50:  2.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497390(CHEMBL3339144)
Affinity DataEC50:  270nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497391(CHEMBL3339147)
Affinity DataEC50:  310nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497392(CHEMBL3339149)
Affinity DataEC50:  4.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497411(CHEMBL3339125)
Affinity DataEC50:  1.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497412(CHEMBL3339122)
Affinity DataEC50:  850nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497413(CHEMBL3339131)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497394(CHEMBL3339136)
Affinity DataEC50:  2.80E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497377(CHEMBL3339142)
Affinity DataEC50:  6.30E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497414(CHEMBL3339145)
Affinity DataEC50:  150nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497419(CHEMBL3339141)
Affinity DataEC50:  2.10E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497378(CHEMBL3339130)
Affinity DataEC50:  490nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50437983(CHEMBL2409106)
Affinity DataEC50:  160nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497421(CHEMBL3339143)
Affinity DataEC50:  3.20E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497393(CHEMBL3339120)
Affinity DataEC50:  440nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497420(CHEMBL3339148)
Affinity DataEC50:  700nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532002(CHEMBL4530409)
Affinity DataEC50:  129nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532003(CHEMBL4475272)
Affinity DataEC50:  631nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532004(CHEMBL4593085)
Affinity DataEC50:  4.47E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532007(CHEMBL4473433)
Affinity DataEC50:  163nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532012(CHEMBL4461542)
Affinity DataEC50:  81nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532013(CHEMBL4549232)
Affinity DataEC50:  116nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532014(CHEMBL4553987)
Affinity DataEC50:  441nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532015(CHEMBL4550753)
Affinity DataEC50: >3.00E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532016(CHEMBL4472955)
Affinity DataEC50: >3.00E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50532017(CHEMBL4529580)
Affinity DataEC50:  241nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
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