Compile Data Set for Download or QSAR
Report error Found 262 Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 4'
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347074(US10202390, Example 29)
Affinity DataIC50: 2nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347062(US10202390, Example 17)
Affinity DataIC50: 2nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347063(US10202390, Example 18)
Affinity DataIC50: 2nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347061(3-(4-(isopropylamino)-5-(1-(tetrahydro-2H-pyran-4-...)
Affinity DataIC50: 2nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613996(CHEMBL5281961)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347058(US10202390, Example 13)
Affinity DataIC50: 3nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347072(3-(5-(1-(3-hydroxy-3-methylbutyl)-1H-pyrazol-4-yl)...)
Affinity DataIC50: 3nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347064(US10202390, Example 19)
Affinity DataIC50: 3nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347067(US10202390, Example 22)
Affinity DataIC50: 4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347073(US10202390, Example 28)
Affinity DataIC50: 5nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347070(US10202390, Example 25)
Affinity DataIC50: 5nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347060(3-(4-(isopropylamino)-5-(4-propyl-1H-1,2,3-triazol...)
Affinity DataIC50: 6nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347056(2-(6-chloropyrazolo[1,5-a]pyrimidin-3-yl)-N-isopro...)
Affinity DataIC50: 8nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50505262(CHEMBL4559408)
Affinity DataKi:  8.20nMAssay Description:Inhibition GIRK1/4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347059(US10202390, Example 14)
Affinity DataIC50: 9nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347057(US10202390, Example 12)
Affinity DataIC50: 9nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM585727(US11530213, Example 48 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347068(US10202390, Example 23)
Affinity DataIC50: 9nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347071(US10202390, Example 26)
Affinity DataIC50: 10nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613997(CHEMBL5280047)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347065(US10202390, Example 20)
Affinity DataIC50: 12nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347066(US10202390, Example 21)
Affinity DataIC50: 14nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347048(US10202390, Example 3)
Affinity DataIC50: 14nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347069(US10202390, Example 24)
Affinity DataIC50: 14nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347051(US10202390, Example 6)
Affinity DataIC50: 18nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347055(US10202390, Example 10)
Affinity DataIC50: 20nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM585709(US11530213, Example 30 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613999(CHEMBL5289977)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347054(US10202390, Example 9)
Affinity DataIC50: 29nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347052(US10202390, Example 8 | US10202390, Example 7)
Affinity DataIC50: 43nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613992(CHEMBL5282689)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347052(US10202390, Example 8 | US10202390, Example 7)
Affinity DataIC50: 53nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347047(2-(7-chloroimidazo[1,2-b]pyridazin-3-yl)-N-isoprop...)
Affinity DataIC50: 63nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM585682(US11530213, Example 3 | 8-chloro-1-(2,6-dichloroph...)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50614001(CHEMBL5278366)
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM585681(US11530213, Example 2 | (R)-8-chloro-1-(2,6- dichl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50614002(CHEMBL5285569)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50437979(CHEMBL2409110)
Affinity DataEC50:  110nMAssay Description:Activation of GIRK1/4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613994(CHEMBL5269440)
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50593405(CHEMBL5178783)
Affinity DataEC50:  145nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM585680(US11530213, Example 1)
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM585699(US11530213, Example 20 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM347050(US10202390, Example 5)
Affinity DataIC50: 174nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50437954(CHEMBL2409269)
Affinity DataIC50: 180nMAssay Description:Inhibition of GIRK1/4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613993(CHEMBL5286246)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50497417(CHEMBL3339101)
Affinity DataIC50: 200nMAssay Description:Inhibition of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613995(CHEMBL5290509)
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50593381(CHEMBL5192713)
Affinity DataEC50:  229nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50439410(CHEMBL2420532)
Affinity DataEC50:  240nMAssay Description:Activation of GIRK1/4 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM585688(US11530213, Example 9 | 8-chloro-1-(2,6-dichloroph...)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
Displayed 1 to 50 (of 262 total ) | Next | Last >>
Jump to: