Compile Data Set for Download or QSAR
Report error Found 259 Enz. Inhib. hit(s) with Target = 'Gastrin-releasing peptide receptor'
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe-...)
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(cyclopropylbenzene(CO)His-Trp-Ala-Val-DAla-His-DPr...)
Affinity DataIC50: 0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040325(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)DPhe...)
Affinity DataIC50: 0.0380nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071733(Compound GRP | CHEMBL413196)
Affinity DataKi:  0.0400nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(cyclopropylbenzene(CO)His-Trp-Ala-Val-DAla-His-DPr...)
Affinity DataIC50: 0.0490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50: 0.0500nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158698([N40,Pro1,Tyr4]BB | CHEMBL266078)
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50275902(D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe-Nle-NH2 | CHEM...)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at recombinant gastrin releasing peptide receptor expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50: 0.0790nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158699([(N4-Bzdig)0]BB(7-14) | CHEMBL414307)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  0.150nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158697([N40,Pro1,Tyr4,Nle 14]BB | CHEMBL268222)
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  0.150nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 0.160nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe-...)
Affinity DataIC50: 0.220nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.230nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataEC50:  0.258nMAssay Description:Displacement of 125I[Tyr4]-bombesin from GRPR expressed in human PC3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50: 0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040320(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Tyr-...)
Affinity DataIC50: 0.330nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50374870(CHEMBL272335)
Affinity DataEC50:  0.373nMAssay Description:Displacement of 125I[Tyr4]-bombesin from GRPR expressed in human PC3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158698([N40,Pro1,Tyr4]BB | CHEMBL266078)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407275(CHEMBL2112786)
Affinity DataIC50: 0.490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50066009(CHEMBL3401466)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I-Tyr4]bombesin from GRPR (unknown origin) expressed in human PC3 cells after 45 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040316(3-isoquinolyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 0.570nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50279041((2S)-N1-((5S,8S,11S,17S,20S,23S,26S,29S,35S,38S)-1...)
Affinity DataIC50: 0.590nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158700([(N4-Bzdig)0,Nle14]BB(7-14) | CHEMBL266079)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50: 0.600nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50066009(CHEMBL3401466)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I-Tyr4]bombesin from GRPR (unknown origin) expressed in human PC3 cells after 45 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158699([(N4-Bzdig)0]BB(7-14) | CHEMBL414307)
Affinity DataIC50: 0.650nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50288252(Bombesin analogue | CHEMBL269432)
Affinity DataKi:  0.700nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071744(AcBB(7-14) | CHEMBL314375)
Affinity DataKi:  0.700nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158702(Universal ligand | CHEMBL413893)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85480(CAS_l | (3-Ph-Pr6)His7,DAla11,DPro13,Psi13-14,Phe1...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040324(PhCH2CH2(CO)His-(BzthAla)-Ala-Val-DAla-His-Pro(psi...)
Affinity DataIC50: 0.75nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85500(Bombesin,Phe13)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158701([Tyr4]Bombesin | CHEMBL407101)
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.990nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50275902(D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe-Nle-NH2 | CHEM...)
Affinity DataKi:  0.990nMAssay Description:Binding affinity to gastrin releasing peptide receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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