Compile Data Set for Download or QSAR
Report error Found 2090 Enz. Inhib. hit(s) with Target = 'Glucagon receptor'
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266669(CHEMBL4093458)
Affinity DataEC50:  5.80E+4nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266670(CHEMBL4065846)
Affinity DataEC50:  5.70E+3nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266671(CHEMBL4101203)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266676(CHEMBL4074468)
Affinity DataEC50:  4.20E+4nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266672(CHEMBL4100420)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266674(CHEMBL4098061)
Affinity DataEC50:  0.0260nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266677(CHEMBL4080035)
Affinity DataEC50:  0.00190nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266675(CHEMBL4090347)
Affinity DataEC50:  0.00890nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266678(CHEMBL4060629)
Affinity DataEC50:  2.32nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266687(CHEMBL4072029)
Affinity DataEC50:  1.24nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266688(CHEMBL4065550)
Affinity DataEC50:  0.00620nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266689(CHEMBL4095024)
Affinity DataEC50:  0.00630nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50241203(exenatide | HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGSPPP...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50152769(GLP-1(7-36)-NH2 | NH2-HAEGTFTSDVSSYLEGQAAKEFIAWLVK...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266690(CHEMBL439305)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266692(CHEMBL4082505)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50152769(GLP-1(7-36)-NH2 | NH2-HAEGTFTSDVSSYLEGQAAKEFIAWLVK...)
Affinity DataEC50: >0.00100nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50241203(exenatide | HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGSPPP...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266668(CHEMBL4098545)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.000400nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266690(CHEMBL439305)
Affinity DataEC50: >0.00100nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266695(CHEMBL4098991)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.00130nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266691(CHEMBL4086979)
Affinity DataEC50:  0.0250nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266673(CHEMBL4076828)
Affinity DataEC50:  1.12nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266694(CHEMBL4069307)
Affinity DataEC50:  0.0160nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266691(CHEMBL4086979)
Affinity DataEC50:  0.000700nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275564(CHEMBL4128125)
Affinity DataEC50:  0.000700nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275567(CHEMBL4128194)
Affinity DataEC50:  0.00160nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275568(CHEMBL4126738)
Affinity DataEC50:  0.0276nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275566(CHEMBL4128276)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275565(CHEMBL4125912)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275595(CHEMBL4127525)
Affinity DataEC50:  0.00190nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275596(CHEMBL4129347)
Affinity DataEC50:  0.00670nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275598(CHEMBL4126027)
Affinity DataEC50:  0.0154nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275545(CHEMBL4126953)
Affinity DataEC50:  0.0276nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275594(CHEMBL4130225)
Affinity DataEC50:  0.00440nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275593(CHEMBL4126812)
Affinity DataEC50:  0.00250nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275546(CHEMBL4130044)
Affinity DataEC50:  42.9nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275569(CHEMBL4130148)
Affinity DataEC50:  3.09nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275578(CHEMBL4128112)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.000500nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50241203(exenatide | HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGSPPP...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50277055(CHEMBL4169653)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50277056(CHEMBL4163714)
Affinity DataEC50:  0.460nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50277057(CHEMBL4174154)
Affinity DataEC50:  0.860nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50277063(CHEMBL4163731)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50277068(CHEMBL4167169)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50277070(CHEMBL4170976)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 2090 total ) | Next | Last >>
Jump to: