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Report error Found 606 Enz. Inhib. hit(s) with Target = 'Heparanase'
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50614394(CHEMBL5273238)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human heparanase using fondaparinux as substrate incubated for 18 hrs by Polymer-H fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50614394(CHEMBL5273238)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of heparanase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388329(CHEMBL2059500)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50611959(CHEMBL5276024)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human heparanase incubated for 4 hrs by beta-scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50466629(CHEMBL4280766)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant HPSE (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388343(CHEMBL2059243)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388341(CHEMBL2059241)
Affinity DataKi:  5.80nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50614397(CHEMBL5279386)
Affinity DataKi:  6nMAssay Description:Binding affinity to heparanase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388342(CHEMBL2059242)
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388331(CHEMBL2059499)
Affinity DataKi:  6.10nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388345(CHEMBL2059245)
Affinity DataKi:  6.40nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50378647(PI-88 | CHEMBL1627122)
Affinity DataKi:  7.90nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388332(CHEMBL2059498)
Affinity DataKi:  8.40nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388346(CHEMBL2059246)
Affinity DataKi:  8.5nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388336(CHEMBL2059504)
Affinity DataKi:  9.10nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388335(CHEMBL2059503)
Affinity DataKi:  9.10nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388330(CHEMBL2059247)
Affinity DataKi:  10.5nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388328(CHEMBL2059505)
Affinity DataKi:  11.3nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50614397(CHEMBL5279386)
Affinity DataIC50: 12nMAssay Description:Inhibition of heparanase (unknown origin) incubated for 18 hrs by fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50612819(CHEMBL5291042)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human HPSE expressed in insect cells by fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50611973(CHEMBL5282692)
Affinity DataIC50: 12nMAssay Description:Inhibition of HPSE (unknown origin) using fondaparinux as substrate incubated for 18 hrs by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388334(CHEMBL2059501)
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50431651(CHEMBL2349236)
Affinity DataIC50: 17nMAssay Description:Inhibition of HPSE (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50093526(CHEMBL426373 | RK-682)
Affinity DataIC50: 17nMAssay Description:Inhibition of HPSE (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50614398(CHEMBL5268939)
Affinity DataIC50: 20nMAssay Description:Inhibition of heparanase (unknown origin) incubated for 18 hrs by fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50611974(CHEMBL5271999)
Affinity DataIC50: 20nMAssay Description:Inhibition of HPSE (unknown origin) using fondaparinux as substrate incubated for 18 hrs by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50612820(CHEMBL5267246)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human HPSE expressed in insect cells by fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388333(CHEMBL2059502)
Affinity DataKi:  20nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640013(CHEMBL5562364)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640011(CHEMBL5559476)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388344(CHEMBL2059244)
Affinity DataKi:  22.3nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640010(CHEMBL5561988)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640009(CHEMBL5549928)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388340(CHEMBL2059510)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640004(CHEMBL5557429)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640007(CHEMBL5556661)
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640012(CHEMBL5557768)
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640006(CHEMBL5559840)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640003(CHEMBL5564261)
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50647174(CHEMBL5597984)
Affinity DataIC50: 57nMAssay Description:Inhibition of HPSE1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50175932(1,3-bis-[4-(5,6-dimethyl-1H-benzoimidazol-2-yl)phe...)
Affinity DataIC50: 75nMAssay Description:Inhibition of recombinant heparanase catalytic stie (unknown origin) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50175932(1,3-bis-[4-(5,6-dimethyl-1H-benzoimidazol-2-yl)phe...)
Affinity DataIC50: 75nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50466636(CHEMBL4286441)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant HPSE (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640005(CHEMBL5560024)
Affinity DataIC50: 82nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640008(CHEMBL5559647)
Affinity DataIC50: 85nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50640002(CHEMBL5561039)
Affinity DataIC50: 92nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50104680(3-Hexadecanoyl-5-hydroxymethyl-4-methoxy-5H-furan-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HPSE (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50611970(CHEMBL5286960)
Affinity DataIC50: 100nMAssay Description:Inhibition of HPSE (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50388338(CHEMBL2059508)
Affinity DataKi:  111nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50618639(CHEMBL5432881)
Affinity DataIC50: 120nMAssay Description:Inhibition of heparanase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
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