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Report error Found 1627 Enz. Inhib. hit(s) with Target = 'Hexokinase-4'
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34101(benzamide derivative, 14e)
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34104(benzamide derivative 15a)
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34102(benzamide derivative 15b)
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34105(benzamide derivative 15c)
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34071(benzamide derivative, 6)
Affinity DataEC50:  67.1nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34072(benzamide derivative, 12)
Affinity DataEC50:  1.26E+4nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34073(benzamide derivative, 13a)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34074(benzamide derivative, 13b)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34075(benzamide derivative, 13c)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34076(benzamide derivative, 13d)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34077(benzamide derivative, 13e)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34078(benzamide derivative, 13f)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34079(benzamide derivative, 13g)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34080(benzamide derivative, 13h)
Affinity DataEC50:  1.87E+3nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34081(benzamide derivative, 13i)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34082(benzamide derivative, 13j)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34083(benzamide derivative, 13k)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34084(benzamide derivative, 13l)
Affinity DataEC50:  2.53E+3nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34085(benzamide derivative, 13m)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34086(benzamide derivative, 13n)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34087(benzamide derivative, 13o)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34088(benzamide derivative, 13p)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34089(benzamide derivative, 13q)
Affinity DataEC50:  2.13E+3nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34090(benzamide derivative, 13r)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34091(benzamide derivative, 13s)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34092(benzamide derivative, 13t)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34093(benzamide derivative, 13u)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34094(benzamide derivative, 13v)
Affinity DataEC50:  1.36E+3nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34095(benzamide derivative, 13w)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34096(benzamide derivative, 13x)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34097(benzamide derivative, 14a)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34098(benzamide derivative, 14b)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34099(benzamide derivative, 14c)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM34100(benzamide derivative, 14d)
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229602(US9340506, A-1)
Affinity DataEC50:  1.40E+3nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229603(US9340506, A-11)
Affinity DataEC50:  950nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229604(US9340506, A-12)
Affinity DataEC50:  660nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229605(US9340506, A-32)
Affinity DataEC50: >1.00E+4nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229606(US9340506, A-58)
Affinity DataEC50: >1.00E+4nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229607(US9340506, B-4)
Affinity DataEC50:  3.70E+3nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229608(US9340506, B-9)
Affinity DataEC50:  93nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM228449(US9556135, 71 | BDBM229609 | US9340506, G3B)
Affinity DataEC50:  1.12E+3nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229610(US9340506, B-20)
Affinity DataEC50:  590nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229611(US9340506, B-23)
Affinity DataEC50:  480nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229612(US9340506, B-26)
Affinity DataEC50:  220nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229613(US9340506, B-49)
Affinity DataEC50:  570nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229614(US9340506, B-58)
Affinity DataEC50:  740nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229615(US9340506, C3)
Affinity DataEC50:  130nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM229616(US9340506, D1)
Affinity DataEC50:  100nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

TargetHexokinase-4(Human)
Shanghai Institutes For Biological Sciences

LigandPNGBDBM228457(US9556135, 102 | BDBM229617 | US9340506, G20A)
Affinity DataEC50:  140nMpH: 7.2Assay Description:The assay is carried out according to the protocol outlined in Hariharan et al (1997), Diabetes 46: 11-16. Briefly, the test compounds are incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
US Patent

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