Compile Data Set for Download or QSAR
Report error Found 8543 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase'
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM50241990(CHEMBL502489 | Camboginol | Garcinol, 1 | Garcinol)
Affinity DataKd:  400nMT: 2°CAssay Description:The p300 activity assays were performed by a colorimetric kit (JM-K322-100, MBL) using active recombinant p300/HAT as positive control and acetyl-CoA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM84873(Nemorosone, 2)
Affinity DataKd:  250nMT: 2°CAssay Description:The p300 activity assays were performed by a colorimetric kit (JM-K322-100, MBL) using active recombinant p300/HAT as positive control and acetyl-CoA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM84874(Guttiferone A, 3)
Affinity DataKd:  100nMT: 2°CAssay Description:The p300 activity assays were performed by a colorimetric kit (JM-K322-100, MBL) using active recombinant p300/HAT as positive control and acetyl-CoA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM84875(Guttiferone E, 4)
Affinity DataKd:  390nMT: 2°CAssay Description:The p300 activity assays were performed by a colorimetric kit (JM-K322-100, MBL) using active recombinant p300/HAT as positive control and acetyl-CoA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM84877(Clusianone, 10)
Affinity DataKd:  810nMT: 2°CAssay Description:The p300 activity assays were performed by a colorimetric kit (JM-K322-100, MBL) using active recombinant p300/HAT as positive control and acetyl-CoA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human PCAF (G715 to D831 residues) expressed in mammalian expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2019
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2019
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataKd:  87nMAssay Description:Binding affinity to human EP300 (A1040 to G1161 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2019
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT8(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-azanylnaphthalen-1-ol;hydrochloride | PCMD-CC-PA...)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT8(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-azanylnaphthalen-1-ol;hydrochloride | PCMD-CC-PA...)
Affinity DataKd:  700nMAssay Description:Binding affinity to N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKd:  110nMAssay Description:Binding affinity to human EP300 (A1040 to G1161 residues) expressed in bacterial expression system by BROMOScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase GCN5(Baker's yeast)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50371146(CHEMBL4168633)
Affinity DataKd:  4.20E+3nMAssay Description:Binding affinity to yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase GCN5(Baker's yeast)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372744(CHEMBL4165080)
Affinity DataKd:  2.62E+4nMAssay Description:Binding affinity to yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM179481(US9675697, Cpd. No. 73)
Affinity DataKd: >4.00E+3nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM179481(US9675697, Cpd. No. 73)
Affinity DataKd:  550nMAssay Description:Binding affinity to human partial length EP300 (A1040 to G1161 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM179481(US9675697, Cpd. No. 73)
Affinity DataKd: >4.00E+3nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM50453949(CHEMBL4208820 | US11247989, Example 87)
Affinity DataKd:  0.120nMAssay Description:Binding affinity to human partial length EP300 (A1040 to G1161 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50453949(CHEMBL4208820 | US11247989, Example 87)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50453949(CHEMBL4208820 | US11247989, Example 87)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged PCAF expressed in mammalian expression system by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM50455480(CHEMBL4218735)
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged EP300 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged GCN5L2 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT8(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50470500(CHEMBL4291334)
Affinity DataKd:  1.90E+4nMAssay Description:Binding affinity to human His-tagged MOF by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Universitá

LigandPNGBDBM249277(US9458145, 1020-18 | US10017501, Compound 1020-18)
Affinity DataKd:  220nMAssay Description:Binding affinity to human partial length EP300 (A1040 to G1161 residues) expressed in bacterial expression system after 1 hr by bromoscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM249277(US9458145, 1020-18 | US10017501, Compound 1020-18)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system after 1 hr by bromoscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM249277(US9458145, 1020-18 | US10017501, Compound 1020-18)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system after 1 hr by bromoscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512955(CHEMBL4454395)
Affinity DataKd:  7.80E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512954(CHEMBL4527339)
Affinity DataKd:  138nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512956(CHEMBL4437954)
Affinity DataKd:  3.04E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512957(CHEMBL4460616)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512963(CHEMBL4475074)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512964(CHEMBL4574669)
Affinity DataKd:  78nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512965(CHEMBL4453637)
Affinity DataKd:  100nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512966(CHEMBL4570924)
Affinity DataKd:  120nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512967(CHEMBL4449143)
Affinity DataKd:  118nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512959(CHEMBL4454766)
Affinity DataKd:  183nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512968(CHEMBL4454700)
Affinity DataKd:  106nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512969(CHEMBL4539318)
Affinity DataKd:  233nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512970(CHEMBL4470046)
Affinity DataKd:  820nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512971(CHEMBL4471746)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512972(CHEMBL4579627)
Affinity DataKd:  621nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512973(CHEMBL4438712)
Affinity DataKd:  1.19E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512974(CHEMBL4471600)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512961(CHEMBL4541223)
Affinity DataKd:  242nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512962(CHEMBL4565832)
Affinity DataKd:  215nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512975(CHEMBL4471748)
Affinity DataKd:  152nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512964(CHEMBL4574669)
Affinity DataKd:  105nMAssay Description:Binding affinity to human N-terminal His-tagged GCN5 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase KAT2B(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50512960(CHEMBL4545594)
Affinity DataKd:  128nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
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