Compile Data Set for Download or QSAR
Report error Found 2505 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 5'
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250182(CHEMBL4077331)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250199(CHEMBL4092477)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)
Affinity DataEC50:  375nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250201(CHEMBL4070639)
Affinity DataEC50:  137nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250202(CHEMBL4074680)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250203(CHEMBL4083755)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250204(CHEMBL4060937)
Affinity DataEC50:  916nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250205(CHEMBL4067491)
Affinity DataEC50:  110nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)
Affinity DataEC50:  635nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250207(CHEMBL4082585)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250208(CHEMBL4062443)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250213(CHEMBL4104927)
Affinity DataEC50:  752nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250210(CHEMBL4087072)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250215(CHEMBL4091536)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250212(CHEMBL4089119)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  34nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250206(CHEMBL4060816)
Affinity DataEC50:  299nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250209(CHEMBL4090425)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250586(CHEMBL4093140)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50026883(CHEMBL437050)
Affinity DataEC50:  550nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50268806(Ac-Tyr-Val-Nle-Gly-His-DPhe-Arg-Trp-Asp-Arg-Phe-Gl...)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250591(CHEMBL4072387)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250585(CHEMBL4104092)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250582(CHEMBL4068654)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250587(CHEMBL4079302)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50258953(CHEMBL4086679)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50258946(CHEMBL4089149)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50258947(CHEMBL4078828)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50258954(CHEMBL4087835)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50258949(CHEMBL4072797)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50263382(CHEMBL4065418)
Affinity DataEC50:  5.20E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50263383(CHEMBL4079142)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50263393(CHEMBL4072638)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50263382(CHEMBL4065418)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50263381(CHEMBL4097903)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50263383(CHEMBL4079142)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266701(CHEMBL4064728)
Affinity DataEC50:  2.60E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266731(CHEMBL4092424)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266702(CHEMBL4102613)
Affinity DataEC50:  5.40E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266732(CHEMBL4084671)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266749(CHEMBL4092849)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266751(CHEMBL4065189)
Affinity DataEC50:  7.20E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266713(CHEMBL4089759)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266714(CHEMBL4068643)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266757(CHEMBL4080138)
Affinity DataEC50:  2.90E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
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